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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T15712 | Laropiprant | MK-0524 | Prostaglandin Receptor |
Laropiprant (MK-0524) is a potent and selective antagonist of prostaglandin D2 (PGD2) receptor (DP) such as and DP/DP1 receptor(Ki = 0.57 nM) and TP Receptor(Ki = 2.95 nM). | |||
T14842 | BW 245C | BW245C | Prostaglandin Receptor |
BW 245C is a selective prostaglandin-like DP receptor (DP1) agonist, a prostaglandin analogue with inhibitory effects on the aggregation response of collagen, which can be used to study diseases such as stroke. | |||
T14148 | AH 6809 | Prostaglandin Receptor | |
AH 6809 is an antagonist of EP and DP receptor(with Kis of 1217, 1150, 1597, and 1415 nM for the cloned human EP1, EP2, EP3-III, and DP receptor respectively). AH 6809 has a Ki of 350 nM for mouse EP2 receptor. | |||
T7359 | CAY10471 Racemate | TM30089 Racemate | GPR , Prostaglandin Receptor |
CAY10471 Racemate (TM30089 Racemate) is a potent, highly selective CRTH2/DP 2 receptor antagonist. CAY10471 Racemate binds to the human CRTH2/DP2, DP1, and TP receptors( Ki values of 0.6, 1200, and >10,000 nM,respectivel... | |||
T4624 | PGD2-IN-1 | PGD2-inhibitor | Prostaglandin Receptor |
PGD2-IN-1 (PGD2-inhibitor) is an effective DP receptor antagonist (IC50:0.3 nM), a compound that can inhibit prostaglandin D2 (PGD2) signaling. PGD2-IN-1 specifically targets and regulates the activity of PGD2 receptors ... | |||
T27765 | L-644,698 | ||
L-644,698 is a selective agonist of human prostanoid DP receptor. | |||
T29225 | ZK118182 isopropyl ester | ZK118182,ZK 118182,ZK-118182 | |
ZK118182 isopropyl ester is a PG analog with potent DP-agonist activity (EC50 = 16.5 nM) and high affinity for the DP receptor (Ki = 74 nM). | |||
T70265 | AL-6556 | ||
AL-6556 is a prostaglandin DP receptor agonist. | |||
T64267 | Laropiprant sodium | ||
Laropiprant sodium is a potent and selective DP receptor antagonist with Ki values of 0.57 nM for TP receptors and 2.95 nM for DP receptors. | |||
T80073 | Dp[Tyr(methyl)2,Arg8]-Vasopressin | Vasopressin Receptor | |
Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1]. | |||
T38113 | AL 6598 | ||
Elevated intraocular pressure (IOP) is an important risk factor in developing glaucoma. Certain prostaglandins such as PGF2α and PGD2, have been shown to reduce IOP. AL 6598 is the isopropyl ester prodrug of AL 6556, a P... | |||
T14146 | AGN 210676 | Simenepag | Prostaglandin Receptor |
AGN 210676 is a selective agonist of prostaglandin EP2(EC50 : 5 nM). | |||
T15828 | L 888607 | Others | |
L 888607 is an effective and selective CRTH2 agonist (Ki: 0.8 nM). |